Triacetin

Basic Information

Name: Triacetin

CAS No: 1,2,3-Propanetriol triacetate [102-76-1]

Functional Categories

Humectant Plasticizer Solvent

1. Nonproprietary Names

BP: Triacetin PhEur: Triacetin USP: Triacetin

2. Synonyms

Captex 500; E1518; glycerol triacetate; glyceryl triacetate; triacetinum; triacetyl glycerine.

3. Chemical Name & CAS Registry

1,2,3-Propanetriol triacetate [102-76-1]

4. Empirical Formula & Molecular Weight

C9H14O6 218.21

5. Structural Formula

6. Applications

Triacetin is mainly used as a hydrophilic plasticizer in both aqueous and solvent-based polymeric coating of capsules, tablets, beads, and granules; typical concentrations used are 10–35% w/w.(1,2) Triacetin is used in cosmetics, perfumery, and foods as a solvent and as a fixative in the formulation of perfumes and flavors.

7. Description

Triacetin is a colorless, viscous liquid with a slightly fatty odor.

8. Pharmacopeial Specifications

See Table I.

9. Typical Properties

Autoignition temperature 4328C Boiling point 2588C Density 1.16 g/cm3 at 258C Explosive limits 1.05% at 1898C lower limit; 7.73% at 2158C upper limit. Flash point 1538C (open cup) Freezing point 3.28C (supercools to about –708C) Melting point 788C Refractive index nD 25 = 1.4296 Solubility see Table II. Vapor density (relative) 7.52 (air = 1) Vapor pressure 133 Pa (1 mmHg) at 1008C Viscosity (dynamic) 1111 mPa s (1111 cP) at –17.88C; 107 mPa s (107 cP) at 08C; 17.4 mPa s (17.4 cP) at 258C; 1.8 mPa s (1.8 cP) at 1008C.

10. Stability & Storage

Triacetin is stable and should be stored in a well-closed, nonmetallic container, in a cool, dry place.

11. Incompatibilities

Triacetin is incompatible with metals and may react with oxidizing agents. Triacetin may destroy rayon fabric.

12. Method of Manufacture

Triacetin is prepared by the esterification of glycerin with acetic anhydride.

13. Safety

Triacetin is used in oral pharmaceutical formulations and is generally regarded as a relatively nontoxic and nonirritant material at the levels employed as an excipient.(3) LD50 (dog, IV): 1.5 g/kg(4) LD50 (mouse, IP): 1.4 g/kg LD50 (mouse, IV): 1.6 g/kg LD50 (mouse, oral): 1.1 g/kg LD50 (mouse, SC): 2.3 g/kg LD50 (rabbit, IV): 0.75 g/kg LD50 (rat, IP): 2.1 g/kg LD50 (rat, oral): 3 g/kg LD50 (rat, SC): 2.8 g/kg

14. Handling Precautions

Observe normal precautions appropriate to the circumstances and quantity of material handled. Triacetin may be irritant to the eyes; eye protection and gloves are recommended.

15. Regulatory Status

GRAS listed. Accepted in Europe as a food additive in certain applications. Included in the FDA Inactive Ingredients Database (oral capsules and tablets and gels). Included in nonparenteral medicines licensed in the UK. Included in the Canadian List of Acceptable Non-medicinal Ingredients.

16. Related Substances

17. Comments

A specification for triacetin is contained in the Food Chemicals Codex (FCC).(5) The EINECS number for triacetin is 203-051-9. The PubChem Compound ID (CID) for triacetin is 5541.